For treatment of prostate cancer, endometriosis, uterine fibroids and premature puberty
Leuprolide binds to the gonadotropin releasing hormone receptor and acts as a potent inhibitor of gonadotropin secretion.
~3 hours
* 27 L [intravenous bolus administration to healthy male volunteers]
* 8.34 L/h [healthy male receiving a 1-mg IV bolus]