TIROSINT

UNIVADIS - TIROSINT /univadis/TIROSINT.md

ATC

Μορφές: SOFT.CAPS

Δραστικές

Δελτίο Τιμών 05/2018

Ημερομηνία barcode code περιεχομενο τιμή παραγωγός χονδρική λιανική
05/2018 2802927401018 292740101 TIROSINT SOFT.CAPS 13MC/CAP BTx30 CAPS 5.47 5.77 8.25
05/2018 2802927402015 292740201 TIROSINT SOFT.CAPS 25MC/CAP BTx30 CAPS 5.47 5.77 8.25
05/2018 2802927403012 292740301 TIROSINT SOFT.CAPS 50MC/CAP BTx30 CAPS 5.47 5.77 8.25
05/2018 2802927404019 292740401 TIROSINT SOFT.CAPS 75MC/CAP BTx30 CAPS 5.47 5.77 8.25
05/2018 2802927405016 292740501 TIROSINT SOFT.CAPS 88MC/CAP BTx30 CAPS 5.53 5.83 8.34
05/2018 2802927406013 292740601 TIROSINT SOFT.CAPS 100MC/CAP BTx30 CAPS 5.53 5.83 8.34
05/2018 2802927407010 292740701 TIROSINT SOFT.CAPS 112MC/CAP BTx30 CAPS 5.53 5.83 8.34
05/2018 2802927408017 292740801 TIROSINT SOFT.CAPS 125MC/CAP BTx30 CAPS 5.53 5.83 8.34
05/2018 2802927409014 292740901 TIROSINT SOFT.CAPS 137MC/CAP BTx30 CAPS 5.61 5.91 8.46
05/2018 2802927410010 292741001 TIROSINT SOFT.CAPS 150MC/CAP BTx30 CAPS 5.61 5.91 8.46
05/2018 2802927411017 292741101 TIROSINT SOFT.CAPS 175MC/CAP BTx30 CAPS 5.61 5.91 8.46
05/2018 2802927412014 292741201 TIROSINT SOFT.CAPS 200MC/CAP BTx30 CAPS 5.61 5.91 8.46
  • DRUGBANK - Levothyroxine
  • indication:

    For use alone or in combination with antithyroid agents to treat hypothyroidism, goiter, chronic lymphocytic thyroiditis, myxedema coma, and stupor.

  • pharmacology:

  • mechanism:

    Levothyroxine acts like the endogenous thyroid hormone thyroxine (T<sub>4</sub>, a tetra-iodinated tyrosine derivative). In the liver and kidney, T<sub>4</sub> is converted to T<sub>3</sub>, the active metabolite. In order to increase solubility, the thyroid hormones attach to thyroid hormone binding proteins, thyroxin-binding globulin, and thyroxin-binding prealbumin (transthyretin). Transport and binding to thyroid hormone receptors in the cytoplasm and nucleus then takes place. Thus by acting as a replacement for natural thyroxine, symptoms of thyroxine deficiency are relieved.

  • toxicity:

    LD<sub>50</sub>=20 mg/kg (orally in rat). Hypermetabolic state indistinguishable from thyrotoxicosis of endogenous origin. Symptoms of thyrotoxicosis include weight loss, increased appetite, palpitations, nervousness, diarrhea, abdominal cramps, sweating, tachycardia, increased pulse and blood pressure, cardiac arrhythmias, tremors, insomnia, heat intolerance, fever, and menstrual irregularities.

  • absorprion:

    Bioavailability varies from 48% to 80%. Human studies have confirmed the importance of an intact jejunum and ileum for levothyroxine absorption and have shown some absorption from the duodenum.

  • halflife:

    T<sub>4</sub>, 6 to 7 days. T<sub>3</sub>, 1 to 2 days.

  • roouteelimination:

    Thyroid hormones are primarily eliminated by the kidneys.

  • volumedistribution:

  • clearance: